Talsifirtosin

A takaice bayanin:

CAS:328898-40

Takaddun shaida:Gmp & iso

Shirya:25kg / Drum

Samfura:Wanda akwai

 

 


Farashin FOB US $ 0.5 - 9,999 / Sashi
Minrimer 1 yanki
Wadatarwa 10000 guda daya a wata
Lokacin biyan kudi T / t, d / p, d / a, l / c

Cikakken Bayani

Bayanan Kamfanin

Tags samfurin

Talsifirtosin

Talsifirosin wani sabon nau'in zobe na Semi-roba macrolorride na dabbobi, wanda shine ainihin tynlosi.

Mataki na magunguna

A kan rigakafin ƙwayoyin cuta na TilIPirosi ya yi kama da na Tylosin, kuma yana da ƙarfi mai haɓaka ƙwararraki akan ƙwayoyin cuta na ƙwayoyin cuta da kuma wasu ƙwayoyin cuta marasa kyau. Tsarin ƙwayoyin cuta na TilIPirosi na TilIPirOSIN daidai yake da na macrolides. Zai iya haɗawa tare da 50s subduit daga cikin ribosome na ƙwayoyin cuta mai mahimmanci don hana syntharia na sunadarai na ƙwayoyin cuta. Tattaunawa na abubuwan da aka gyara guda biyu na musamman da Tillifiros ya bambanta da tsarin wannan magani daga Tylosin da tilpodin, inda aka sanya 20-piperIDine a cikin lumen don tsoma baki tare da ci gaban nascent peptides.

Saboda tediroxine yana da ƙungiyoyi 3 na Amino na asali, ana iya samar da siffofin caji daban-daban a ƙarƙashin yanayin PH. Adadin cajin shine babban mahimmancin tushen abubuwan ƙwayoyin cuta na ƙwayoyin cuta kuma ya shiga ciki membrane na ƙwayoyin cuta, don haka ƙwayoyin cuta mara kyau na Tillipirosin a cikin vitro an kwashe shi da ph. A karkashin yanayin acidic, ana haifar da ƙungiyar amino, sakamakon a cikin raguwa a cikin ayyukan rigakafin ƙwayoyin cuta na tediroxine, yayin da a cikin yanayin alkaline na ƙwayoyin cuta.

Macrologies infita m cytokanes, aikin phospholipase, da kuma sakin liyafa, kuma suna da tasirin anti-mai kumburi a cikin Macrophage da neutrophils. Tediroxine yana rage barna mai kumburi a lokacin wasu kumburi ko martani.

Kwayar otitback

Tildipirosin is effective against pathogenic bacteria that cause respiratory diseases in pigs and cattle (such as Pasteurella multocida, Actinobacillus pleuropneumoniae, Bordetella bronchiseptica, Haemophilus parasuis, Mannheim spp. etc.) the antibacterial activity of tilmicosin was 2-32 times higher than that of tilmicosin, Kuma ayyukan ƙwayoyin rigakafin ƙwayoyin rigakafin ƙwayoyin cuta sun yi fissiichia Coli sun fi Tylosin da Tilmomosin. Hakanan yana kula da wasu nau'ikan Mycoplasma, Sprachees, Relcella na binciken kwayar cuta ta HAEMophilus akan Pleuropnesico. Tillifirosin shine kwayar cuta ga wasu ƙwayoyin cuta (kamar haemophilus parasuis da Attenobacnopnese )e), yayin da yake yawanci ƙwayoyin cuta (kamar shi ne Motatocia (kamar shi a PastecoLla Mercocida). Don ƙwayoyin cuta na ciki, tare da rage darajar PH (daga 7.3 zuwa 6.3 zuwa 64), Mic na Tillipirosidis da Escherichia Coripirtois na Salmonel / M zuwa 64 ~ ml. Saboda haka, sakamakon canje-canje na PH a Vivo ya kamata a yi la'akari lokacin da gudanar da gwajin gwajin cutar kantunan Toripirtosin. Bugu da kari, Mic na Tillipirsin da Motarfin Pastecolla Motako ne 0.5ug / ml a cikin Serum, wanda ya kasance da alaƙa da wannan lokacin.

Inococus-Streptococcus a cikin shanu shanu suna da tsayayya da tediroxine. Tillifiros ne mai zaman kansa ga Multocida da Mannheimia Haemolyticus dauke da gentes. Hakanan, yanayin da aka lalata da shi na M. Bovis yana da tsayayya wa rigakafin rigakafin macrolorride ciki har da Tillipirosin. Wasu raunin HAEMophilus parasuis an kuma samu su kasance a zahiri da tediroxine. Mycoplasma Bovis iya hanzarin juriya ga Tillipirosin, amma saboda jinkirin ci gaban mycoplasma, a cikin gwajin kwantar da hankali na iya jinkirta magani. Nazari ya nuna cewa yankin II (nucleotide 748) da kuma yanki v (maye gurbi a cikin nucleotides 2059 da 2060) suna da alaƙa da ƙara yawan juriya ga macrolides. Sabili da haka, mai saukin kamuwa da M. Bovis zuwa magunguna na Macrolide da sauri ta gwajin wannan maye gurbi.

Tiamulin-hydrogen-fumate1

Wadatacce

98%

Gwadawa

Tsarin Kamfanin


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